505982 (-)-Quinpirole Hydrochloride - CAS 85798-08-9 - Calbiochem

MSDS (material safety data sheet) or SDS, CoA and CoQ, dossiers, brochures and other available documents.

Synonyms: Dopamine D₂ Receptor Agonist, Quinpirole, Quinpirole, LY-171,555, LY 171555

Primary Target: D₂
505982
Price could not be retrieved
Minimum Quantity needs to be mulitiple of
Upon Order Completion More Information
You Saved ()
 
—
Request Pricing
—
Limited AvailabilityLimited Availability
Stocked 
Discontinued
Limited Quantities Available
Available
    Remaining : Will advise
      Remaining : Will advise
      Will advise
      Contact Customer Service
      Contact Customer Service
      View Pricing & Availability

      Overview

      Replacement Information

      Key Specifications Table

      Empirical FormulaCAS #
      C₁₃H₂₁N₃•HCl 85798-08-9

      Pricing & Availability

      Catalog Number AvailabilityPackaging Qty/Pack Price Quantity
      5.05982.0001
      Retrieving availability...
      —
      Limited AvailabilityLimited Availability
      Stocked 
      Discontinued
      Limited Quantities Available
      Available
        Remaining : Will advise
          Remaining : Will advise
          Will advise
          Contact Customer Service
          Contact Customer Service

          		 Glass bottle 10 mg
          Retrieving price...
          Price could not be retrieved
          Minimum Quantity needs to be mulitiple of
          Upon Order Completion More Information
          You Saved ()
           
          —
          Request Pricing
          		 —
          Description
          OverviewA potent, selective dopamine D2 receptor agonist with a Ki value of 4.8 nM. Some D3(Ki = 24 nM) and D4 (Ki = 30 nM) receptor agonistic action has also been reported. In rat striatum studies in vitro, application of quinpriole inhibited single pulse dopamine overflow in a concentration-dependent manner (IC50 = 32.5 nM).
          Catalogue Number505982
          Brand Family Calbiochem®
          SynonymsDopamine D₂ Receptor Agonist, Quinpirole, Quinpirole, LY-171,555, LY 171555
          References
          ReferencesOʹNeill, C. et al. 2009. J. Neurochem. 108, 545.
          Malmberg, A. and Mohell, N. 1995. J. Pharmacol. Exp. Ther. 274, 790.
          Seeman, P. and Schaus, J. M. 1991. Eur. J. Pharmacol. 203, 105.
          Product Information
          CAS number85798-08-9
          FormWhite powder
          Hill FormulaC₁₃H₂₁N₃•HCl
          Chemical formulaC₁₃H₂₁N₃•HCl
          Structure formula ImageStructure formula Image
          Applications
          Biological Information
          Primary TargetD₂
          Primary Target K<sub>i</sub>4.8 nM
          Purity≥98% by HPLC
          Physicochemical Information
          Dimensions
          Materials Information
          Toxicological Information
          Safety Information according to GHS
          Safety Information
          Product Usage Statements
          Storage and Shipping Information
          Ship Code Shipped at Ambient Temperature or with Blue Ice or with Dry Ice
          Toxicity Standard Handling
          Storage -20°C
          Protect from Light Protect from light
          Do not freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
          Packaging Information
          Transport Information
          Supplemental Information
          Specifications

          Documentation

          (-)-Quinpirole Hydrochloride - CAS 85798-08-9 - Calbiochem SDS

          Title

          Safety Data Sheet (SDS) 

          References

          Reference overview
          OʹNeill, C. et al. 2009. J. Neurochem. 108, 545.
          Malmberg, A. and Mohell, N. 1995. J. Pharmacol. Exp. Ther. 274, 790.
          Seeman, P. and Schaus, J. M. 1991. Eur. J. Pharmacol. 203, 105.
          Data Sheet

          Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

          Revision12-September-2013 JSW
          SynonymsDopamine D₂ Receptor Agonist, Quinpirole, Quinpirole, LY-171,555, LY 171555
          DescriptionA potent, selective dopamine D2 receptor agonist with a Ki value of 4.8 nM. Some D3(Ki = 24 nM) and D4 (Ki = 30 nM) receptor agonistic action has also been reported. In rat striatum studies in vitro, application of quinpriole inhibited single pulse dopamine overflow in a concentration-dependent manner (IC50 = 32.5 nM).
          FormWhite powder
          CAS number85798-08-9
          Chemical formulaC₁₃H₂₁N₃•HCl
          Structure formulaStructure formula
          Purity≥98% by HPLC
          SolubilityH₂O (7.3 mg/ml)
          Storage -20°C
          Protect from light
          Do Not Freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
          Toxicity Standard Handling
          ReferencesOʹNeill, C. et al. 2009. J. Neurochem. 108, 545.
          Malmberg, A. and Mohell, N. 1995. J. Pharmacol. Exp. Ther. 274, 790.
          Seeman, P. and Schaus, J. M. 1991. Eur. J. Pharmacol. 203, 105.