505894 | CGP 7930 - CAS 57717-80-3 - Calbiochem

505894
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      Overview

      Replacement Information

      Key Specifications Table

      Empirical FormulaCAS #
      C₁₉H₃₂O₂ 57717-80-3

      Pricing & Availability

      Catalog NumberAvailability Packaging Qty/Pack Price Quantity
      5.05894.0001
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          Glass bottle 10 mg
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          Description
          OverviewA blood brain barrier permeable, positive allosteric modulator of the metabotropic GABAB receptor. Shown to modulate GABAB receptor in the high affinity state and thereby increases agonist affinity for the receptor. Also enhances agonist potency and efficacy even on recombinant GABAB receptors. Exhibits anxiolytic effects in rodents.
          Catalogue Number505894
          Brand Family Calbiochem®
          SynonymsGABA B Receptor Antagonist, CGP7930, CGP 7930, CGP-7930
          References
          ReferencesAdams, C. et al., 2007. CNS Drug Rev. 13, 308.
          Pin, J.P., et al., 2007. Curr. Neuropharmacol. 5, 195.
          Product Information
          CAS number57717-80-3
          FormPale yellow solid
          Hill FormulaC₁₉H₃₂O₂
          Chemical formulaC₁₉H₃₂O₂
          Structure formula ImageStructure formula Image
          Applications
          Biological Information
          Primary TargetGABAB
          Purity≥98% by HPLC
          Physicochemical Information
          Dimensions
          Materials Information
          Toxicological Information
          Safety Information according to GHS
          Safety Information
          Product Usage Statements
          Storage and Shipping Information
          Ship Code Shipped at Ambient Temperature or with Blue Ice or with Dry Ice
          Toxicity Standard Handling
          Storage +2°C to +8°C
          Protect from Light Protect from light
          Do not freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
          Packaging Information
          Transport Information
          Supplemental Information
          Specifications

          Documentation

          SDS

          Title

          Safety Data Sheet (SDS) 

          References

          Reference overview
          Adams, C. et al., 2007. CNS Drug Rev. 13, 308.
          Pin, J.P., et al., 2007. Curr. Neuropharmacol. 5, 195.
          Data Sheet

          Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

          Revision20-September-2013 JSW
          SynonymsGABA B Receptor Antagonist, CGP7930, CGP 7930, CGP-7930
          DescriptionA blood brain barrier permeable, positive allosteric modulator of the metabotropic GABAB receptor. Shown to modulate GABAB receptor in the high affinity state and thereby increases agonist affinity for the receptor. Also enhances agonist potency and efficacy even on recombinant GABAB receptors. Exhibits anxiolytic effects in rodents.
          FormPale yellow solid
          CAS number57717-80-3
          Chemical formulaC₁₉H₃₂O₂
          Structure formulaStructure formula
          Purity≥98% by HPLC
          SolubilityDMSO (100 mM) or Ethanol (100 mM)
          Storage +2°C to +8°C
          Protect from light
          Do Not Freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
          Toxicity Standard Handling
          ReferencesAdams, C. et al., 2007. CNS Drug Rev. 13, 308.
          Pin, J.P., et al., 2007. Curr. Neuropharmacol. 5, 195.