504795 | BRL 44408 Maleate - CAS 118343-19-4 - Calbiochem

504795
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      Overview

      Replacement Information

      Key Specifications Table

      Empirical FormulaCAS #
      C₁₃H₁₇N₃ • C₄H₄O₄ 118343-19-4

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      5.04795.0001
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          Glass bottle 10 mg
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          Description
          OverviewA selective α2A-adrenoceptor antagonist (Ki = 1.7 nM and 144.5 nM at α2A and α2B-adrenergic receptors respectively). Has been used to study regulation of neurotransmitter release from sympathetic nerves and shown to increase hippocampal noradrenaline release following systemic administration.
          Catalogue Number504795
          Brand Family Calbiochem®
          Synonyms2-[(4,5-Dihydro-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-methyl-1H-isoindole maleate
          References
          ReferencesAlberts, P., et al. 1993. General Pharmacology 24, 1.
          Imaki, J., et al. 2009. Neuroscience Letters 454, 143.
          Carlos, M., et al. 2012. Eur. J. Pharmacol. 683, 204.
          Product Information
          CAS number118343-19-4
          FormTan powder
          Hill FormulaC₁₃H₁₇N₃ • C₄H₄O₄
          Chemical formulaC₁₃H₁₇N₃ • C₄H₄O₄
          Hygroscopic Hygroscopic
          Structure formula ImageStructure formula Image
          Applications
          Biological Information
          Primary Target2A-adrenoceptor
          Primary Target K<sub>i</sub>1.7 nM and 144.5 nM at →2A and →2B-adrenergic receptors respectively
          Purity≥98% by HPLC
          Physicochemical Information
          Dimensions
          Materials Information
          Toxicological Information
          Safety Information according to GHS
          Safety Information
          Product Usage Statements
          Storage and Shipping Information
          Ship Code Shipped at Ambient Temperature or with Blue Ice or with Dry Ice
          Toxicity Standard Handling
          Storage -20°C
          Protect from Light Protect from light
          Protect from Moisture Protect from moisture
          Hygroscopic Hygroscopic
          Do not freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
          Packaging Information
          Transport Information
          Supplemental Information
          Specifications

          Documentation

          SDS

          Title

          Safety Data Sheet (SDS) 

          References

          Reference overview
          Alberts, P., et al. 1993. General Pharmacology 24, 1.
          Imaki, J., et al. 2009. Neuroscience Letters 454, 143.
          Carlos, M., et al. 2012. Eur. J. Pharmacol. 683, 204.
          Data Sheet

          Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

          Revision12-July-2013 JSW
          Synonyms2-[(4,5-Dihydro-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-methyl-1H-isoindole maleate
          DescriptionA selective ?2A-adrenoceptor antagonist (Ki = 1.7 nM and 144.5 nM at ?2A and ?2B-adrenergic receptors respectively). Has been used to study regulation of neurotransmitter release from sympathetic nerves and shown to increase hippocampal noradrenaline release following systemic administration.
          FormTan powder
          CAS number118343-19-4
          Chemical formulaC₁₃H₁₇N₃ • C₄H₄O₄
          Structure formulaStructure formula
          Purity≥98% by HPLC
          SolubilityH₂O (10 mg/ml)
          Storage -20°C
          Hygroscopic
          Protect from moisture
          Protect from light
          Do Not Freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
          Toxicity Standard Handling
          ReferencesAlberts, P., et al. 1993. General Pharmacology 24, 1.
          Imaki, J., et al. 2009. Neuroscience Letters 454, 143.
          Carlos, M., et al. 2012. Eur. J. Pharmacol. 683, 204.