539560 PKC Inhibitor Peptide 19-36

539560
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      Overview

      Replacement Information

      Key Specifications Table

      Empirical Formula
      C₉₃H₁₅₉N₃₅O₂₄

      Pricing & Availability

      Catalog Number AvailabilityPackaging Qty/Pack Price Quantity
      539560-500UG
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          Plastic ampoule 500 μg
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          Description
          OverviewActs as pseudosubstrate by binding to the active sites of protein kinase C. A potent, reversible, and substrate competitive inhibitor of protein kinase C (Ki = 147 nM) but not of protein kinase A (IC50 = 423 µM).
          Catalogue Number539560
          Brand Family Calbiochem®
          SynonymsProtein Kinase C Inhibitor Peptide 19-36, RFARKGALRQKNVHEVKN
          References
          ReferencesMakowske, M. and Rosen, O.M. 1989. J. Biol. Chem. 264, 16155.
          House, C. and Kemp, B.E. 1987. Science 238, 1726.
          Product Information
          ATP CompetitiveN
          FormWhite to off-white lyophilized solid
          FormulationSupplied as a trifluoroacetate salt.
          Hill FormulaC₉₃H₁₅₉N₃₅O₂₄
          Chemical formulaC₉₃H₁₅₉N₃₅O₂₄
          Hygroscopic Hygroscopic
          ReversibleY
          Sold on the basis of peptide contentY
          Applications
          Biological Information
          Primary TargetPKC
          Primary Target K<sub>i</sub>147 nM against protein kinase C
          Purity≥95% by HPLC
          Physicochemical Information
          Cell permeableN
          Peptide ContentY
          Peptide SequenceH-Arg-Phe-Ala-Arg-Lys-Gly-Ala-Leu-Arg-Gln-Lys-Asn-Val-His-Glu-Val-Lys-Asn-OH
          Dimensions
          Materials Information
          Toxicological Information
          Safety Information according to GHS
          Safety Information
          Product Usage Statements
          Storage and Shipping Information
          Ship Code Ambient Temperature Only
          Toxicity Standard Handling
          Storage -20°C
          Hygroscopic Hygroscopic
          Do not freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 4 weeks at -20°C.
          Packaging Information
          Transport Information
          Supplemental Information
          Specifications

          Documentation

          PKC Inhibitor Peptide 19-36 SDS

          Title

          Safety Data Sheet (SDS) 

          PKC Inhibitor Peptide 19-36 Certificates of Analysis

          TitleLot Number
          539560

          References

          Reference overview
          Makowske, M. and Rosen, O.M. 1989. J. Biol. Chem. 264, 16155.
          House, C. and Kemp, B.E. 1987. Science 238, 1726.
          Data Sheet

          Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

          Revision11-January-2010 RFH
          SynonymsProtein Kinase C Inhibitor Peptide 19-36, RFARKGALRQKNVHEVKN
          DescriptionActs as pseudosubstrate by binding to the active sites of protein kinase C. A potent, reversible, and substrate competitive inhibitor of protein kinase C (Ki = 147 nM) but not of protein kinase A (IC50 = 423 µM).
          FormWhite to off-white lyophilized solid
          FormulationSupplied as a trifluoroacetate salt.
          Chemical formulaC₉₃H₁₅₉N₃₅O₂₄
          Peptide SequenceH-Arg-Phe-Ala-Arg-Lys-Gly-Ala-Leu-Arg-Gln-Lys-Asn-Val-His-Glu-Val-Lys-Asn-OH
          Purity≥95% by HPLC
          SolubilityH₂O (0.1%)
          Storage -20°C
          Hygroscopic
          Do Not Freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 4 weeks at -20°C.
          Toxicity Standard Handling
          ReferencesMakowske, M. and Rosen, O.M. 1989. J. Biol. Chem. 264, 16155.
          House, C. and Kemp, B.E. 1987. Science 238, 1726.