361555 | GSK-3 Inhibitor XIII - CAS 404828-08-6 - Calbiochem

361555
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      Overview

      Replacement Information

      Key Specifications Table

      Empirical FormulaCAS #
      C₁₈H₁₅N₅ 404828-08-6

      Pricing & Availability

      Catalog NumberAvailability Packaging Qty/Pack Price Quantity
      361555-1MG
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          Plastic ampoule 1 mg
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          361555-5MG
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              Description
              OverviewAn aminopyrazole compound that acts as a potent and ATP-binding site inhibitor of GSK-3 with a Ki of 24 nM.
              Catalogue Number361555
              Brand Family Calbiochem®
              Synonyms(5-Methyl-1H-pyrazol-3-yl)-(2-phenylquinazolin-4-yl)amine
              References
              ReferencesPierce, A.C., et al. 2005. J. Med. Chem. 48, 1278.
              Product Information
              CAS number404828-08-6
              ATP CompetitiveN
              FormWhite solid
              Hill FormulaC₁₈H₁₅N₅
              Chemical formulaC₁₈H₁₅N₅
              ReversibleN
              Structure formula ImageStructure formula Image
              Applications
              Biological Information
              Primary TargetGSK-3
              Primary Target K<sub>i</sub>24 nM against GSK-3
              Purity≥95% by HPLC
              Physicochemical Information
              Cell permeableN
              Dimensions
              Materials Information
              Toxicological Information
              Safety Information according to GHS
              Safety Information
              Product Usage Statements
              Storage and Shipping Information
              Ship Code Ambient Temperature Only
              Toxicity Carcinogenic / Teratogenic
              Storage +2°C to +8°C
              Protect from Light Protect from light
              Do not freeze Ok to freeze
              Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
              Packaging Information
              Transport Information
              Supplemental Information
              Specifications

              Documentation

              SDS

              Title

              Safety Data Sheet (SDS) 

              Certificates of Analysis

              TitleLot Number
              361555

              References

              Reference overview
              Pierce, A.C., et al. 2005. J. Med. Chem. 48, 1278.

              Brochure

              Title
              Calbiochem Biologics 32.1
              Data Sheet

              Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

              Revision01-July-2008 RFH
              Synonyms(5-Methyl-1H-pyrazol-3-yl)-(2-phenylquinazolin-4-yl)amine
              DescriptionA potent and ATP-competitive inhibitor of GSK-3 (Ki = 24 nM).
              FormWhite solid
              CAS number404828-08-6
              Chemical formulaC₁₈H₁₅N₅
              Structure formulaStructure formula
              Purity≥95% by HPLC
              SolubilityDMSO (5 mg/ml)
              Storage +2°C to +8°C
              Protect from light
              Do Not Freeze Ok to freeze
              Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
              Toxicity Carcinogenic / Teratogenic
              ReferencesPierce, A.C., et al. 2005. J. Med. Chem. 48, 1278.