371780 | GP Antagonist-2A - Calbiochem

371780
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      Overview

      Replacement Information

      Key Specifications Table

      Empirical Formula
      C₇₉H₁₀₅N₂₁O₁₃S

      Pricing & Availability

      Catalog NumberAvailability Packaging Qty/Pack Price Quantity
      371780-1MG
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          Plastic ampoule 1 mg
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          Description
          OverviewA peptide that selectively inhibits the activation of Gq by M1-muscarinic cholinergic receptors. Also inhibits activation by cholecystokinin receptor in pancreatic acini at 10 µM. Blocks angiotensin II-stimulated sis-inducing factor and STAT3 tyrosine phosphorylation.
          Catalogue Number371780
          Brand Family Calbiochem®
          SynonymsRPKPQQDWFDWDWM
          References
          ReferencesHunt, R.A., et al. 1999. Hypertension 34, 603.
          Tsunoda Y., et al. 1995. Biochem. Biophys. Res. Commun. 211, 648.
          Mukai, H., et al. 1992. J. Biol. Chem. 267, 16237.
          Product Information
          ATP CompetitiveN
          FormLyophilized solid
          FormulationSupplied as a trifluoroacetate salt.
          Hill FormulaC₇₉H₁₀₅N₂₁O₁₃S
          Chemical formulaC₇₉H₁₀₅N₂₁O₁₃S
          ReversibleN
          Applications
          Biological Information
          Primary TargetInhibits the activation of Gq by M1-muscarinic cholinergic receptors
          Purity≥95% by HPLC
          Physicochemical Information
          Cell permeableN
          Peptide SequenceH-Arg-Pro-Lys-Pro-Gln-Gln-D-Trp-Phe-D-Trp-D-Trp-Met-NH₂
          Dimensions
          Materials Information
          Toxicological Information
          Safety Information according to GHS
          Safety Information
          Product Usage Statements
          Storage and Shipping Information
          Ship Code Ambient Temperature Only
          Toxicity Standard Handling
          Storage -20°C
          Do not freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 1 month at -20°C.
          Packaging Information
          Transport Information
          Supplemental Information
          Specifications

          Documentation

          SDS

          Title

          Safety Data Sheet (SDS) 

          Certificates of Analysis

          TitleLot Number
          371780

          References

          Reference overview
          Hunt, R.A., et al. 1999. Hypertension 34, 603.
          Tsunoda Y., et al. 1995. Biochem. Biophys. Res. Commun. 211, 648.
          Mukai, H., et al. 1992. J. Biol. Chem. 267, 16237.
          Data Sheet

          Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

          Revision13-May-2010 JSW
          SynonymsRPKPQQDWFDWDWM
          DescriptionA peptide that selectively inhibits the activation of Gq by M1-muscarinic cholinergic receptors. Also inhibits activation by cholecystokinin receptor in pancreatic acini at 10 µM. Blocks angiotensin II-stimulated sis-inducing factor and STAT3 tyrosine phosphorylation.
          FormLyophilized solid
          FormulationSupplied as a trifluoroacetate salt.
          Chemical formulaC₇₉H₁₀₅N₂₁O₁₃S
          Peptide SequenceH-Arg-Pro-Lys-Pro-Gln-Gln-D-Trp-Phe-D-Trp-D-Trp-Met-NH₂
          Purity≥95% by HPLC
          SolubilityH₂O (25 mg/ml)
          Storage -20°C
          Do Not Freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 1 month at -20°C.
          Toxicity Standard Handling
          ReferencesHunt, R.A., et al. 1999. Hypertension 34, 603.
          Tsunoda Y., et al. 1995. Biochem. Biophys. Res. Commun. 211, 648.
          Mukai, H., et al. 1992. J. Biol. Chem. 267, 16237.